|
Tabela 2. Unakrsna reaktivnost glavnih metabolita Sirolimusa |
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|
Metabolit |
Bioaktivnost % 336 × 280 |
Koncentracija srodnika do roditelja (%) |
Seimens |
Syva |
Abbott |
|
39-O-demethyl |
10 |
7 |
52% @ |
38% @ |
20.3% @ |
|
16-O-demethyl |
NS |
4 |
10% @ |
15% @ |
7.6% @ |
|
12 hydroxyl |
7 |
11 |
46% @ |
4% @ |
36.8% @ |
|
27, 39-O-didemethyl |
NS |
31 |
89% @ |
52% @ |
NS |
|
Skraćenice : NS, nije navedeno; ACMIA, affinity column-mediated immunoassay; EMIT, enzyme-multiplied immunoassay; and MEIA, microparticle enzyme immunoassay. |
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Tabela 2. Unakrsna reaktivnost glavnih metabolita Sirolimusa Metabolit Bioaktivnost % 7, 8 Koncentracija srodnika do roditelja (%) Seimens ACMIA Syva EMIT Abbott MEIA 39-O-demethyl (41-O-demethyl) 10 7 52% @ 0 ng/mL 60% @ 12 ng/mL 38% @ […]
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